The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
28076824 |
6 |
Discovery of new nanomolar inhibitors of GPa: Extension of 2-oxo-1,2-dihydropyridinyl-3-yl amide-based GPa inhibitors. |
Griffith University |
27522507 |
14 |
Synthetic, enzyme kinetic, and protein crystallographic studies of C-ß-d-glucopyranosyl pyrroles and imidazoles reveal and explain low nanomolar inhibition of human liver glycogen phosphorylase. |
University of Thessaly |
27624527 |
19 |
Synthesis of (benzimidazol-2-yl)aniline derivatives as glycogen phosphorylase inhibitors. |
Egypt National Research Centre |
26851835 |
15 |
2-Oxo-1,2-dihydropyridinyl-3-yl amide-based GPa inhibitors: Design, synthesis and structure-activity relationship study. |
Griffith University |
26713107 |
11 |
4(5)-Aryl-2-C-glucopyranosyl-imidazoles as New Nanomolar Glucose Analogue Inhibitors of Glycogen Phosphorylase. |
University of Debrecen |
26708111 |
41 |
Glucose-derived spiro-isoxazolines are anti-hyperglycemic agents against type 2 diabetes through glycogen phosphorylase inhibition. |
Universit£ |
25092521 |
50 |
Structure based inhibitor design targeting glycogen phosphorylase B. Virtual screening, synthesis, biochemical and biological assessment of novel N-acyl-ß-d-glucopyranosylamines. |
University of Thessaly |
24608000 |
27 |
New synthesis of 3-(ß-D-glucopyranosyl)-5-substituted-1,2,4-triazoles, nanomolar inhibitors of glycogen phosphorylase. |
University of Debrecen |
9406599 |
51 |
A strategy for the incorporation of water molecules present in a ligand binding site into a three-dimensional quantitative structure--activity relationship analysis. |
University of Alcala |
23938052 |
15 |
Synthesis, enzyme kinetics and computational evaluation of N-(ß-D-glucopyranosyl) oxadiazolecarboxamides as glycogen phosphorylase inhibitors. |
University of Debrecen |
24900719 |
12 |
C-Glucopyranosyl-1,2,4-triazoles As New Potent Inhibitors of Glycogen Phosphorylase. |
University of Debrecen |
23395662 |
2 |
Synthesis of tartaric acid analogues of FR258900 and their evaluation as glycogen phosphorylase inhibitors. |
University of Debrecen |
22770609 |
11 |
The binding of C5-alkynyl and alkylfurano[2,3-d]pyrimidine glucopyranonucleosides to glycogen phosphorylase b: synthesis, biochemical and biological assessment. |
University of Thessaly |
22229710 |
18 |
Binding evaluation of fragment-based scaffolds for probing allosteric enzymes. |
Universit£ |
20430629 |
10 |
1-(3-Deoxy-3-fluoro-beta-d-glucopyranosyl) pyrimidine derivatives as inhibitors of glycogen phosphorylase b: Kinetic, crystallographic and modelling studies. |
National Hellenic Research Foundation |
19889536 |
29 |
Terpenoids. III: Synthesis and biological evaluation of 23-hydroxybetulinic acid derivatives as novel inhibitors of glycogen phosphorylase. |
China Pharmaceutical University |
18847277 |
5 |
Practical synthesis of bredemolic acid, a natural inhibitor of glycogen phosphorylase. |
China Pharmaceutical University |
16546381 |
25 |
Pentacyclic triterpenes. Part 3: Synthesis and biological evaluation of oleanolic acid derivatives as novel inhibitors of glycogen phosphorylase. |
China Pharmaceutical University |
16169219 |
6 |
Pentacyclic triterpenes. Part 1: the first examples of naturally occurring pentacyclic triterpenes as a new class of inhibitors of glycogen phosphorylases. |
China Pharmaceutical University |
16143521 |
27 |
Synthesis and evaluation of 3-anilino-quinoxalinones as glycogen phosphorylase inhibitors. |
Johnson & Johnson Pharmaceutical Research and Development |
15214781 |
30 |
Identification, synthesis, and characterization of new glycogen phosphorylase inhibitors binding to the allosteric AMP site. |
Novo Nordisk |
10360741 |
10 |
Efficient inhibition of muscle and liver glycogen phosphorylases by a new glucopyranosylidene-spiro-thiohydantoin. |
Lajos Kossuth University |
22325154 |
25 |
N-(4-Substituted-benzoyl)-N'-(ß-d-glucopyranosyl)ureas as inhibitors of glycogen phosphorylase: Synthesis and evaluation by kinetic, crystallographic, and molecular modelling methods. |
University of Debrecen |
22204907 |
4 |
Design and synthesis of novel photoaffinity probes for study of the target proteins of oleanolic acid. |
China Pharmaceutical University |
21821421 |
8 |
Halogen-substituted (C-ß-D-glucopyranosyl)-hydroquinone regioisomers: synthesis, enzymatic evaluation and their binding to glycogen phosphorylase. |
National Hellenic Research Foundation |
21788139 |
43 |
Ligand-based modelling followed by synthetic exploration unveil novel glycogen phosphorylase inhibitory leads. |
Applied Science University |
21439694 |
161 |
Identification of pentacyclic triterpenes derivatives as potent inhibitors against glycogen phosphorylase based on 3D-QSAR studies. |
Chinese Academy of Sciences |
21123066 |
9 |
Efficient synthesis and biological evaluation of epiceanothic acid and related compounds. |
China Pharmaceutical University |
20947361 |
16 |
The binding ofß-d-glucopyranosyl-thiosemicarbazone derivatives to glycogen phosphorylase: A new class of inhibitors. |
National Hellenic Research Foundation |
19642687 |
36 |
Synthesis of 3-deoxypentacyclic triterpene derivatives as inhibitors of glycogen phosphorylase. |
China Pharmaceutical University |
20080412 |
29 |
Synthesis of 1-(D-glucopyranosyl)-1,2,3-triazoles and their evaluation as glycogen phosphorylase inhibitors. |
University of Debrecen |
19703777 |
12 |
Synthesis and glycogen phosphorylase inhibitory activity of N-(beta-D-glucopyranosyl)amides possessing 1,4-benzodioxane moiety. |
University of Debrecen |
19450985 |
27 |
Synthesis and structure-activity relationships of C-glycosylated oxadiazoles as inhibitors of glycogen phosphorylase. |
University of Debrecen |
19574053 |
9 |
Glucose-based spiro-heterocycles as potent inhibitors of glycogen phosphorylase. |
University of Debrecen |
19348494 |
73 |
Fructose-1,6-bisphosphatase inhibitors. 1. Purine phosphonic acids as novel AMP mimics. |
Metabasis Therapeutics |
18793852 |
14 |
Novel design principle validated: glucopyranosylidene-spiro-oxathiazole as new nanomolar inhibitor of glycogen phosphorylase, potential antidiabetic agent. |
University of Debrecen |
18485716 |
5 |
Evaluation of novel hyphodermin derivatives as glycogen phosphorylase a inhibitors. |
Griffith University |
16970395 |
14 |
Iminosugars as potential inhibitors of glycogenolysis: structural insights into the molecular basis of glycogen phosphorylase inhibition. |
The National Hellenic Research Foundation |
16246555 |
24 |
Pentacyclic triterpenes. Part 2: Synthesis and biological evaluation of maslinic acid derivatives as glycogen phosphorylase inhibitors. |
China Pharmaceutical University |
14643331 |
71 |
Novel 3,4-dihydroquinolin-2(1H)-one inhibitors of human glycogen phosphorylase a. |
Merck Research Laboratories |
14592521 |
50 |
A new class of glycogen phosphorylase inhibitors. |
Merck Research Laboratories |
14505637 |
40 |
Glucose-lowering in a db/db mouse model by dihydropyridine diacid glycogen phosphorylase inhibitors. |
Merck Research Laboratories |
25062009 |
12 |
Synthesis, screening and docking of small heterocycles as glycogen phosphorylase inhibitors. |
Griffith University |
25009003 |
10 |
Glucopyranosylidene-spiro-iminothiazolidinone, a new bicyclic ring system: synthesis, derivatization, and evaluation for inhibition of glycogen phosphorylase by enzyme kinetic and crystallographic methods. |
University of Debrecen |
29453094 |
19 |
A multidisciplinary study of 3-(?-d-glucopyranosyl)-5-substituted-1,2,4-triazole derivatives as glycogen phosphorylase inhibitors: Computation, synthesis, crystallography and kinetics reveal new potent inhibitors. |
University of Debrecen |
28925695 |
25 |
Nanomolar Inhibitors of Glycogen Phosphorylase Based on?-d-Glucosaminyl Heterocycles: A Combined Synthetic, Enzyme Kinetic, and Protein Crystallography Study. |
University of Debrecen |
24119242 |
17 |
Synthesis and evaluation of novel oleanolic acid derivatives as potential antidiabetic agents. |
Chengde Medical University |
19443226 |
10 |
Glycogen phosphorylase inhibitory effects of 2-oxo-1,2-dihydropyridin-3-yl amide derivatives. |
Griffith University |
19781947 |
5 |
Glucose-based spiro-isoxazolines: a new family of potent glycogen phosphorylase inhibitors. |
Universite De Lyon |
19758809 |
66 |
Benzamide derivatives as dual-action hypoglycemic agents that inhibit glycogen phosphorylase and activate glucokinase. |
Shanghai Institutes For Biological Sciences |
18517260 |
26 |
Naturally Occurring Pentacyclic Triterpenes as Inhibitors of Glycogen Phosphorylase: Synthesis, Structure-Activity Relationships, and X-ray Crystallographic Studies. |
China Pharmaceutical University |